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Corrigendum to “Challenges in the development of an M4 PAM preclinical candidate: The discovery, SAR, and biological characterization of a series of azetidine-derived tertiary amides” [Bioorg. Med. Chem. Lett. 27(23) (2017) 5179–5184]

Tarr, James C. ; Wood, Michael R. ; Noetzel, Meredith J. ; [et al.]

Elsevier BV ; 2018

In: Bioorganic & Medicinal Chemistry Letters Vol. 28, No. 17 ( 2018-09), p. 3014-

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In: Bioorganic & Medicinal Chemistry Letters, Elsevier BV, Vol. 28, No. 17 ( 2018-09), p. 3014-

Type of Medium: Online Resource

ISSN: 0960-894X

URL: Article

DOI: 10.1016/j.bmcl.2018.07.022

RVK:

VA 2620

Language: English

Publisher: Elsevier BV

Publication Date: 2018

detail.hit.zdb_id: 1501505-1

SSG: 15,3

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2

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Optimization of M 4 positive allosteric modulators (PAMs): The discovery of VU0476406, a non-human primate in vivo tool compound for translational pharmacology

Melancon, Bruce J. ; Wood, Michael R. ; Noetzel, Meredith J. ; [et al.]

Elsevier BV ; 2017

In: Bioorganic & Medicinal Chemistry Letters Vol. 27, No. 11 ( 2017-06), p. 2296-2301

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In: Bioorganic & Medicinal Chemistry Letters, Elsevier BV, Vol. 27, No. 11 ( 2017-06), p. 2296-2301

Type of Medium: Online Resource

ISSN: 0960-894X

URL: Article

DOI: 10.1016/j.bmcl.2017.04.043

RVK:

VA 2620

Language: English

Publisher: Elsevier BV

Publication Date: 2017

detail.hit.zdb_id: 1501505-1

SSG: 15,3

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3

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Selective Activation of M 4 Muscarinic Acetylcholine Receptors Reverses MK-801-Induced Behavioral Impairments and Enhances Associative Learning in Rodents

Bubser, Michael ; Bridges, Thomas M. ; Dencker, Ditte ; [et al.]

American Chemical Society (ACS) ; 2014

In: ACS Chemical Neuroscience Vol. 5, No. 10 ( 2014-10-15), p. 920-942

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In: ACS Chemical Neuroscience, American Chemical Society (ACS), Vol. 5, No. 10 ( 2014-10-15), p. 920-942

Type of Medium: Online Resource

ISSN: 1948-7193 , 1948-7193

URL: Article

DOI: 10.1021/cn500128b

Language: English

Publisher: American Chemical Society (ACS)

Publication Date: 2014

detail.hit.zdb_id: 2528493-9

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4

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Design of 4-Oxo-1-aryl-1,4-dihydroquinoline-3-carboxamides as Selective Negative Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 2

Felts, Andrew S. ; Rodriguez, Alice L. ; Smith, Katrina A. ; [et al.]

American Chemical Society (ACS) ; 2015

In: Journal of Medicinal Chemistry Vol. 58, No. 22 ( 2015-11-25), p. 9027-9040

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In: Journal of Medicinal Chemistry, American Chemical Society (ACS), Vol. 58, No. 22 ( 2015-11-25), p. 9027-9040

Type of Medium: Online Resource

ISSN: 0022-2623 , 1520-4804

URL: Article

DOI: 10.1021/acs.jmedchem.5b01371

Language: English

Publisher: American Chemical Society (ACS)

Publication Date: 2015

detail.hit.zdb_id: 1491411-6

SSG: 15,3

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5

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Challenges in the development of an M 4 PAM preclinical candidate: The discovery, SAR, and biological characterization of a series of azetidine-derived tertiary amides

Tarr, James C. ; Wood, Michael R. ; Noetzel, Meredith J. ; [et al.]

Elsevier BV ; 2017

In: Bioorganic & Medicinal Chemistry Letters Vol. 27, No. 23 ( 2017-12), p. 5179-5184

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In: Bioorganic & Medicinal Chemistry Letters, Elsevier BV, Vol. 27, No. 23 ( 2017-12), p. 5179-5184

Type of Medium: Online Resource

ISSN: 0960-894X

URL: Article

DOI: 10.1016/j.bmcl.2017.10.053

RVK:

VA 2620

Language: English

Publisher: Elsevier BV

Publication Date: 2017

detail.hit.zdb_id: 1501505-1

SSG: 15,3

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6

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Challenges in the development of an M 4 PAM preclinical candidate: The discovery, SAR, and in vivo characterization of a series of 3-aminoazetidine-derived amides

Tarr, James C. ; Wood, Michael R. ; Noetzel, Meredith J. ; [et al.]

Elsevier BV ; 2017

In: Bioorganic & Medicinal Chemistry Letters Vol. 27, No. 13 ( 2017-07), p. 2990-2995

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In: Bioorganic & Medicinal Chemistry Letters, Elsevier BV, Vol. 27, No. 13 ( 2017-07), p. 2990-2995

Type of Medium: Online Resource

ISSN: 0960-894X

URL: Article

DOI: 10.1016/j.bmcl.2017.05.014

RVK:

VA 2620

Language: English

Publisher: Elsevier BV

Publication Date: 2017

detail.hit.zdb_id: 1501505-1

SSG: 15,3

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7

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A Screen of Approved Drugs Identifies the Androgen Receptor Antagonist Flutamide and Its Pharmacologically Active Metabolite 2-Hydroxy-Flutamide as Heterotropic Activators of Cytochrome P450 3A In Vitro and In Vivo

Blobaum, Anna L. ; Byers, Frank W. ; Bridges, Thomas M. ; [et al.]

American Society for Pharmacology & Experimental Therapeutics (ASPET) ; 2015

In: Drug Metabolism and Disposition Vol. 43, No. 11 ( 2015-11), p. 1718-1726

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In: Drug Metabolism and Disposition, American Society for Pharmacology & Experimental Therapeutics (ASPET), Vol. 43, No. 11 ( 2015-11), p. 1718-1726

Type of Medium: Online Resource

ISSN: 0090-9556 , 1521-009X

URL: Article

DOI: 10.1124/dmd.115.064006

Language: English

Publisher: American Society for Pharmacology & Experimental Therapeutics (ASPET)

Publication Date: 2015

detail.hit.zdb_id: 1500213-5

SSG: 15,3

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8

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Development of Novel, CNS Penetrant Positive Allosteric Modulators for the Metabotropic Glutamate Receptor Subtype 1 (mGlu 1 ), Based on an N -(3-Chloro-4-(1,3-dioxoisoindolin-2-yl)phenyl)-3-methylfuran-2-carboxamide Scaffold, That Potentiate Wild Type and Mutant mGlu 1 Receptors Found in Schizophrenics

Garcia-Barrantes, Pedro M. ; Cho, Hyekyung P. ; Niswender, Colleen M. ; [et al.]

American Chemical Society (ACS) ; 2015

In: Journal of Medicinal Chemistry Vol. 58, No. 20 ( 2015-10-22), p. 7959-7971

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In: Journal of Medicinal Chemistry, American Chemical Society (ACS), Vol. 58, No. 20 ( 2015-10-22), p. 7959-7971

Type of Medium: Online Resource

ISSN: 0022-2623 , 1520-4804

URL: Article

DOI: 10.1021/acs.jmedchem.5b00727

Language: English

Publisher: American Chemical Society (ACS)

Publication Date: 2015

detail.hit.zdb_id: 1491411-6

SSG: 15,3

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9

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Partial mGlu5 Negative Allosteric Modulators Attenuate Cocaine-Mediated Behaviors and Lack Psychotomimetic-Like Effects

Gould, Robert W ; Amato, Russell J ; Bubser, Michael ; [et al.]

Springer Science and Business Media LLC ; 2016

In: Neuropsychopharmacology Vol. 41, No. 4 ( 2016-3), p. 1166-1178

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In: Neuropsychopharmacology, Springer Science and Business Media LLC, Vol. 41, No. 4 ( 2016-3), p. 1166-1178

Type of Medium: Online Resource

ISSN: 0893-133X , 1740-634X

URL: Article

DOI: 10.1038/npp.2015.265

RVK:

WA 15000

Language: English

Publisher: Springer Science and Business Media LLC

Publication Date: 2016

detail.hit.zdb_id: 2008300-2

SSG: 15,3

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10

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Heterotropic Activation of the Midazolam Hydroxylase Activity of CYP3A by a Positive Allosteric Modulator of mGlu 5 : In Vitro to In Vivo Translation and Potential Impact on Clinically Relevant Drug-Drug Interactions

Blobaum, Anna L. ; Bridges, Thomas M. ; Byers, Frank W. ; [et al.]

American Society for Pharmacology & Experimental Therapeutics (ASPET) ; 2013

In: Drug Metabolism and Disposition Vol. 41, No. 12 ( 2013-12), p. 2066-2075

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In: Drug Metabolism and Disposition, American Society for Pharmacology & Experimental Therapeutics (ASPET), Vol. 41, No. 12 ( 2013-12), p. 2066-2075

Type of Medium: Online Resource

ISSN: 0090-9556 , 1521-009X

URL: Article

DOI: 10.1124/dmd.113.052662

Language: English

Publisher: American Society for Pharmacology & Experimental Therapeutics (ASPET)

Publication Date: 2013

detail.hit.zdb_id: 1500213-5

SSG: 15,3

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