In:
Journal of Heterocyclic Chemistry, Wiley, Vol. 54, No. 1 ( 2017-01), p. 325-330
Abstract:
A series of novel 1‐(3‐chloropyridin‐2‐yl)‐ N ‐substituted‐5‐(trifluoromethyl)‐pyrazole carboxamide derivatives TC 1 , TC 2 , TC 3 , TC 4 , TC 5 , TC 6 , TC 7 , TC 8 , TC 9 , TC 10 , TC 11 were synthesized and characterized by IR, 1 H NMR, 13 C NMR, MS, and elemental analysis. All the target compounds were tested in vitro for their antibacterial activities and antifungal activities. The preliminary bioassays indicated that compound TC 6 exhibited excellent activity against Xanthomonas oryzae (94.9% and 84.9%) at different concentrations (200 µg/mL and 100 µg/mL), which was higher than that of Bismerthiazol (94.6% and 64.0%), respectively. At the same time, most of the compounds exhibited moderate antifungal activities against four kinds of phytopathogenic fungi
Type of Medium:
Online Resource
ISSN:
0022-152X
,
1943-5193
Language:
English
Publisher:
Wiley
Publication Date:
2017
detail.hit.zdb_id:
2042274-X
Bookmarklink