In:
Advanced Synthesis & Catalysis, Wiley, Vol. 359, No. 3 ( 2017-02-02), p. 390-394
Abstract:
The first efficient regioselective pyridylation of 1‐ tert ‐butoxycarbonyl‐3‐iodoazetidine to produce 2‐ and 3‐heteroarylazetidines under palladium‐catalyzed conditions has been developed. The established direct pyridylation of azetidines affords 2‐ vs . 3‐heteroarylazetidines in moderate to good yields (up to 92%) and with good regioselectivity (up to 98:2) by using different ligands. magnified image
Type of Medium:
Online Resource
ISSN:
1615-4150
,
1615-4169
DOI:
10.1002/adsc.201600470
Language:
English
Publisher:
Wiley
Publication Date:
2017
detail.hit.zdb_id:
2041384-1
detail.hit.zdb_id:
2033084-4