In:
European Journal of Organic Chemistry, Wiley, Vol. 2017, No. 37 ( 2017-10-10), p. 5671-5678
Abstract:
A para ‐toluenesulfonic acid ( p TSA) catalyzed domino aza‐Piancatelli rearrangement/Michael reaction was developed for the construction of 1,4‐benzodiazepin‐5‐ones in one pot. The method proceeds well in the presence of various furfurylcarbinols and o ‐aminobenzamides to give products that contain medicinally relevant chemical entities.
Type of Medium:
Online Resource
ISSN:
1434-193X
,
1099-0690
DOI:
10.1002/ejoc.v2017.37
DOI:
10.1002/ejoc.201700957
Language:
English
Publisher:
Wiley
Publication Date:
2017
detail.hit.zdb_id:
1475010-7