Format:
1 Online-Ressource
ISBN:
9783527674404
,
3527674381
,
3527674411
,
9783527674381
,
9783527674411
Series Statement:
Methods and principles in medicinal chemistry vol. 72
Content:
Introduction. Polypharmacology in Drug Discovery / Oscar Méndez-Lucio, J Jesús Naveja, Hugo Vite-Caritino, Fernando D Prieto-Martínez, José L Medina-Franco -- Selectivity of Marketed Drugs. Kinase Inhibitors / Peng Wu, Michael Givskov, Thomas E Nielsen -- Repositioning of Drug - New Indications for Marketed Drugs / Ren Kong, Stephen T Wong -- Discovery Technologies for Drug Repurposing / Naiem T Issa, Stephen W Byers, Sivanesan Dakshanamurthy -- Unselective Drugs in Drug Discovery. Personalized Medicine / Christian Noe, Volker Baumann -- Drug Discovery Strategies for the Generation of Multitarget Ligands against Neglected Tropical Diseases / Annachiara Gandini, Federica Prati, Elisa Uliassi, Maria L Bolognesi -- Designing Approaches to Multitarget Drugs / Luca Costantino, Daniela Barlocco -- The Linker Approach / Daniel Merk, Manfred Schubert-Zsilavecz -- Merged Multiple Ligands / Hongming Chen, Udo Bauer, Ola Engkvist -- Pharmacophore Generation for Multiple Ligands / Norbert Handler -- Cellular Assays / Ye Fang -- Therapeutic Areas for Designed Multiple Ligands. Developing Serotonergic Antidepressants Acting on More Than the Serotonin Transporter / Gerard J Marek -- Multiple Ligands Targeting the Angiotensin System for Hypertension / Agustin Casimiro-Garcia -- Multiple Peroxisome Proliferator-Activated Receptor-Based Ligands / Dmytro Kukhtar, Miquel Mulero, Raul Beltrán-Debón, Cristina Valls, Gerard Pujadas, Santiago Garcia-Vallve -- Antibiotics / Jean-Philippe Surivet, Philippe Panchaud -- Multiple Ligands in Neurodegenerative Diseases / Julien Lalut, Christophe Rochais, Patrick Dallemagne
Additional Edition:
9783527335381
Additional Edition:
Erscheint auch als Druck-Ausgabe Drug selectivity Weinheim : Wiley-VCH Verlag & Co. KGaA, 2018 3527335382
Additional Edition:
9783527335381
Language:
English
Subjects:
Chemistry/Pharmacy
Keywords:
Arzneimittelforschung
;
Individualisierte Medizin
DOI:
10.1002/9783527674381
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